Ibhanti kunye nendlela: Intsebenziswano, uVumelwano kunye nokuphumelela phakathi koBuntu
iimveliso

Iimveliso

I-Delamanid CAS: 681492-22-8

I-Delamanid liyeza elilwa ne-mycobacterial elichazwa njenge-diarylquinoline derivative, elisetyenziswa kakhulu kunyango lwe-multidrug-resistant tuberculosis (MDR-TB). Isebenza ngokujolisa kwi-mycobacterial ATP synthase, ekhokelela ekuphazamisekeni kwemveliso yamandla kwiibhaktheriya ezibangela isifo sephepha. I-Delamanid ithathwa njengearhente yodidi lwesibini kwiimeko ze-MDR-TB apho kukho ukuxhathisa kumayeza okuqala aqhelekileyo. Eli yeza lifumaneka kwifom yethebhulethi kwaye lidla ngokumiselwa njengenxalenye yerejimeni epheleleyo yokulwa nosulelo lwesifo sephepha oluchasene namayeza.


Iinkcukacha zeMveliso

Iithegi zeMveliso

Ukusetyenziswa kunye nesiphumo:

I-Delamanid sisixhobo esibalulekileyo se-pharmacological ekulawuleni isifo sephepha esinganyangekiyo ngamayeza amaninzi, uhlobo olubi lwesifo sephepha olungaphenduliyo kunyango oluqhelekileyo lomgca wokuqala. Idla ngokubandakanywa kwiindlela zonyango ezidibeneyo ze-MDR-TB ukuphucula iziphumo zonyango kunye nokunciphisa umngcipheko wokukhula kokunganyangeki ngamayeza. Ababoneleli bezempilo banika i-delamanid kunye namanye amayeza omgca wesibini okulwa nesifo sephepha ngokusekelwe kwizinto zesigulana ngasinye, kubandakanya ubungakanani bokunganyangeki ngamayeza, imbali yonyango lwangaphambili, kunye nemeko yempilo iyonke. Amayeza adla ngokusetyenziswa ngomlomo kwifom yethebhulethi, kunye nokuphindaphinda kwedosi kunye nobude bexesha elilungiselelwe iimfuno zesigulana ngasinye. Izigulana ezifumana unyango lwe-delamanid ziyacetyiswa ukuba zilandele ngokungqongqo irejimeni emiselweyo, njengoko ukuthatha amayeza rhoqo kubalulekile ekufezekiseni impumelelo yonyango kunye nokunciphisa umngcipheko wokungaphumeleli konyango. Ukujonga rhoqo iziphumo ebezingalindelekanga, ezinje ngokuphazamiseka kwesisu okanye utshintsho ekusebenzeni kwesibindi, kubalulekile ngexesha lonyango. Unyango lwe-Delamanid ludla ngokuqaliswa kwaye lujongwe ziingcali zempilo ezinamava ekulawuleni iimeko zesifo sephepha esinganyangekiyo ngamayeza. Intsebenziswano phakathi kweqela lezempilo kunye nesigulana ibalulekile ukuqinisekisa ukuthotyelwa konyango, ukujonga inkqubela phambili, kunye nokujongana nazo naziphi na iingxaki okanye iingxaki ngokukhawuleza. Ukuqukumbela, i-delamanid idlala indima ebalulekileyo ekulweni nesifo sephepha esinganyangekiyo ngamayeza amaninzi, inika izigulana kunye nababoneleli bezempilo ukhetho olusebenzayo lokulwa nesi sifo sinzima esosulelayo kunye nokuthintela ukusasazeka kwaso ngakumbi kuluntu.

Isampulu yeMveliso:

I-L-Arginine1
I-L-Arginine2

Ukupakisha imveliso:

I-L-Arginin3

Iinkcukacha ezongezelelweyo:

Ukwakhiwa C25H25F3N4O6
Uvavanyo 99%
Inkangeleko umgubo omhlophe
Inombolo ye-CAS 681492-22-8
Ukupakisha Encinci kwaye ininzi
Beka ubomi kwishelufa iminyaka eyi-2
Indawo yokugcina izinto Gcina kwindawo epholileyo neyomileyo
Isiqinisekiso I-ISO.

 


  • Ngaphambili:
  • Okulandelayo:

  • Bhala umyalezo wakho apha uze uwuthumele kuthi