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I-Somatostatin CAS:51110-01-1
I-Somatostatin yi-hormone yendalo ethintela ukukhululwa kwezinye ii-hormone ezahlukeneyo emzimbeni. Idlala indima ebalulekileyo ekulawuleni inkqubo ye-endocrine kwaye ibandakanyeka ekulawuleni i-hormone yokukhula, i-insulin, i-glucagon, kunye nezinye ii-hormone zesisu.
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I-Linaclotide CAS: 851199-59-2
I-Linaclotide yi-guanylate cyclase-C agonist esetyenziselwa unyango lwe-chronic constipation kunye ne-irritable bowel syndrome kunye ne-constipation kubantu abadala. Isebenza ngaphakathi kwindlela yesisu ukwandisa ukukhutshwa kolwelo kunye nokukhawulezisa ukuhamba kwamathumbu, ukunciphisa iimpawu ezinxulumene nezi meko.
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I-Levosimendan CAS:141505-33-1
I-Levosimendan sisivuseleli se-calcium kunye nesivuli se-potassium channel esisetyenziselwa ukulawula ukusilela kwentliziyo okukhawulezileyo. Eli yeza linefuthe lokunganyibiliki kunye nokuvaleka kwemithambo yegazi, liphucula ukusebenza kwentliziyo kwaye lithomalalise iimpawu zokusilela kwentliziyo.
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I-Liraglutide CAS:204656-20-2
I-Liraglutide liyeza elisetyenziselwa ukunyanga isifo seswekile sohlobo lwesibini kunye nokutyeba kakhulu. Likwiqela lamayeza aziwa ngokuba yi-glucagon-like peptide-1 (GLP-1) receptor agonists, asebenza ngokunyusa imveliso ye-insulin kunye nokunciphisa inani leswekile eveliswa sisibindi. I-Liraglutide ifumaneka ngendlela yokutofa kwaye idla ngokusetyenziswa kanye ngemini. Eli yeza libonakalisiwe ukuba linceda ekunciphiseni amanqanaba eswekile yegazi kwaye likhuthaza ukwehla kobunzima kubantu abanesifo seswekile sohlobo lwesibini kunye nokutyeba kakhulu.
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I-Octreotide Acetate CAS: 83150-76-9
I-Octreotide acetate yi-synthetic octapeptide analog yehomoni yendalo i-somatostatin. Isebenza njengesithinteli esinamandla seehomoni ezahlukeneyo kunye nee-neuropeptides, kwaye isetyenziswa ekulawuleni iimeko ezifana ne-acromegaly, i-carcinoid syndrome, kunye neentlobo ezithile zeethumba.
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I-Semaglutide CAS:910463-68-2
I-Semaglutide yi-glucagon-like peptide-1 (GLP-1) receptor agonist esetyenziselwa ukulawula isifo seswekile sohlobo lwesibini kunye nokutyeba kakhulu. Isebenza ngokulawula amanqanaba eswekile egazini, ukukhuthaza ukwehla kobunzima, kunye nokunciphisa umngcipheko wentliziyo.
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I-Icatibant Acetate CAS:138614-30-9
I-Icatibant acetate liyeza elisetyenziselwa unyango lwe-angioedema yelifa (HAE), imeko engaqhelekanga yemfuza ebonakaliswa kukudumba okukhawulezileyo nokuqatha kolusu, ii-membranes ze-mucous, kunye nezinye izicwili zomzimba. Liyi-bradykinin B2 receptor antagonist ekhethiweyo esebenza ngokuthintela iziphumo ze-bradykinin, umlamli ophambili wokudumba okunxulunyaniswa ne-HAE. I-Icatibant acetate inikwa ngenaliti engaphantsi kwesikhumba kwaye yenzelwe ukunciphisa ngokukhawuleza iimpawu zokuhlaselwa yi-HAE ngokukhawuleza.
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I-Ganirelix Acetate CAS: 123246-29-7
I-Ganirelix acetate liyeza elisetyenziswa kubuchwepheshe bokuncedisa ekuzaleni ukuthintela ukukhutshwa kweqanda ngaphambi kwexesha kubasetyhini abaphantsi kolawulo lwe-ovarian hyperstimulation. Ngokuthintela ukukhululwa kwe-luteinizing hormone, i-ganirelix acetate inceda ekuthinteleni ukukhutshwa kweqanda kwangoko kwaye ixhasa ixesha elifanelekileyo lokufunyanwa kweqanda ngexesha leenkqubo zokuchumisa i-in vitro (IVF). Inikwa nge-subcutaneous injections kwaye idlala indima ebalulekileyo ekulawuleni ngempumelelo unyango lokungazali.
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I-Linaclotide CAS: 851199-59-2
I-Linaclotide sisiyobisi sonyango esisetyenziselwa ukunyanga i-irritable bowel syndrome kunye ne-constipation (IBS-C) kunye ne-chronic idiopathic constipation. Njenge-agonist ye-guanylate cyclase-C, i-linaclotide isebenza ngaphakathi kwindlela yokugaya ukutya ukwandisa ukukhutshwa kolwelo kunye nokukhawulezisa ukuhamba kwamathumbu, ngaloo ndlela inciphisa iimpawu ezifana ne-constipation kunye nokungonwabi kwesisu.
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I-Ziconotide Acetate CAS:107452-89-1
I-Ziconotide acetate yinguqulelo eyenziweyo ye-peptide compound ethathwe kwityhefu ye-Conus magus snail. Isetyenziswa njengeyeza lokuthomalalisa iintlungu ezingapheliyo kwizigulana ezinganyamezelaniyo okanye ezingasabelanga kwezinye iindlela zonyango. I-Ziconotide acetate inikwa ngokufakwa ngaphakathi kwe-thecal, inika isiqabu esijolise kubantu abanengxaki yentlungu engapheliyo.
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I-Degarelix CAS:214766-78-6
I-Degarelix yi-gonadotropin-releasing hormone (GnRH) receptor antagonist esetyenziswa kunyango lomhlaza we-prostate oqhubele phambili. Isebenza ngokucinezela ngokukhawuleza ukuveliswa kwe-testosterone, i-hormone ekhuthaza ukukhula kweethumba ze-prostate.
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I-Acetyl Octapeptide-3/1 CAS:868844-74-0
I-Acetyl Octapeptide-3, ekwaziwa ngokuba yi-Argireline, yi-peptide yokwenziwa esetyenziswa kakhulu kwiimveliso zokhathalelo lolusu ngenxa yeempawu zayo zokulwa nokwaluphala. Kukholelwa ukuba le peptide isebenza ngokunciphisa ukushwabana kwemisipha, nto leyo enokunceda ekunciphiseni ukubonakala kwemigca emincinci kunye nemibimbi, ngakumbi kwiindawo ezinomdla wokubonakala kwemigca efana nebunzi kunye neengqonge amehlo.
