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IPristinamycin CAS:270076-60-3
IPristinamycin liyeza elidibeneyo le-antibiotic eliqulethe izinto ezimbini ezisebenzayo, i-pristinamycin I kunye ne-pristinamycin II. Likwiqela le-streptogramin le-antibiotics kwaye libonisa imisebenzi ye-bacteriostatic kunye ne-bactericidal ngokuchasene neebhaktheriya ezahlukeneyo zegram-positive, kubandakanya i-Staphylococcus aureus kunye ne-Streptococcus pneumoniae. IPristinamycin isebenza ngokuthintela ukwenziwa kweproteni yebhaktheriya, okwenza ukuba isebenze kakuhle ekunyangeni usulelo lolusu kunye nezicubu ezithambileyo, usulelo lwendlela yokuphefumla, kunye nezinye usulelo lwebhaktheriya olubangelwa zizinto eziphilayo ezisengozini.
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I-Ribostamycin sulfate CAS: 53797-35-6
I-Ribostamycin sulfate sisibulali-ntsholongwane se-aminoglycoside esithathwe kwi-Streptomyces griseoluteus. Ibonisa umsebenzi onamandla wokubulala iintsholongwane ngokuchasene neentlobo ezahlukeneyo zeentsholongwane ezine-gram-negative kunye nezinye ezine-gram-positive ngokuthintela ukwenziwa kweproteni. I-Ribostamycin sulfate isetyenziswa kakhulu kunyango lwezifo ezahlukeneyo, kubandakanya izifo zomchamo, izifo zomchamo, izifo zolusu kunye nezicubu ezithambileyo, kunye ne-septicemia ebangelwa ziintsholongwane ezisengozini.
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I-Rifampicin CAS:13292-46-1
I-Rifampicin, eyaziwa ngokuba yi-rifampin, liyeza elibanzi le-antibiotic elikwiqela le-rifamycin. Lisetyenziswa kakhulu kunyango lwesifo sephepha, iqhenqa, kunye nezinye izifo zebhaktheriya. I-Rifampicin isebenza ngokuthintela ukwenziwa kwe-RNA kwiibhaktheriya, ngaloo ndlela iphazamisa amandla azo okuzala nokusinda. Ngenxa yomsebenzi wayo onamandla wokulwa neentsholongwane kunye nokusebenza kakuhle kwiintlobo ze-mycobacterial, i-rifampicin yinxalenye ebalulekileyo yeendlela zonyango ezidibeneyo zesifo sephepha kunye nezinye izifo ezosulelayo.
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I-Puromycin dihydrochloride CAS:58-58-2
I-Puromycin dihydrochloride sisithinteli esinamandla sokwenziwa kwee-antibiotic kunye neeproteni esivela kwi-Streptomyces alboniger. Isetyenziswa kakhulu kuphando lwebhayoloji yeemolekyuli ukuthintela ngokukhethekileyo ukwenziwa kweeproteni kwiiseli ngokuphelisa uguqulelo ngaphambi kwexesha ngexesha lokwenziwa kweeproteni. I-Puromycin dihydrochloride ifakwe kwiitsheyini zepeptide ezisandula ukuzalwa, nto leyo ekhokelela ekukhutshweni kwee-polypeptides ezingaphelelanga kwaye ekugqibeleni ukufa kweeseli. Ngenxa yendlela yayo yokusebenza eyahlukileyo, i-puromycin dihydrochloride sisixhobo esibalulekileyo sokufunda ukwenziwa kweeproteni, umsebenzi we-ribosome, ukubonakaliswa kwezakhi zofuzo, kunye nokuphila kweeseli kwiimeko zovavanyo.
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I-Protionamide CAS:14222-60-7
I-Protionamide liyeza lokubulala iintsholongwane elikwiqela le-thioamide, elisetyenziswa kakhulu kunyango lwesifo sofuba esinganyangekiyo ngamayeza amaninzi. Isebenza ngokuthintela ukwenziwa kwe-mycolic acid eludongeni lweseli yebhaktheriya, nto leyo ekhokelela ekutshatyalalisweni kwesifo sofuba seMycobacterium. I-Protionamide idla ngokumiselwa kunye namanye amayeza okulwa nesifo sofuba njengenxalenye yonyango olupheleleyo lweentlobo zesifo sofuba ezinganyangekiyo ngamayeza.
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I-Potassium clavulanate CAS: 61177-45-5
I-Potassium clavulanate sisithinteli se-β-lactamase esidla ngokudityaniswa nee-antibiotics ezithile ukuphucula ukusebenza kwazo ngokuchasene nosulelo lwebhaktiriya. Isebenza ngokuthintela ukonakala kwe-antibiotic yi-enzymes yebhaktiriya, ngaloo ndlela yandisa uluhlu lomsebenzi kwaye iphucula iziphumo zonyango. I-Potassium clavulanate isetyenziswa rhoqo kwiimveliso ezidibeneyo kunye nee-antibiotics ezifana ne-amoxicillin ukunyanga iintlobo ngeentlobo zosulelo lwebhaktiriya.
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I-Retapamulin CAS:224452-66-8
I-Retapamulin liyeza lokubulala iintsholongwane elikwiqela leziyobisi ze-pleuromutilin. Lisetyenziselwa ukunyanga usulelo lwesikhumba olubangelwa ziintsholongwane, ingakumbi i-impetigo ebangelwa ziintlobo ezibuthathaka ze-Staphylococcus aureus kunye ne-Streptococcus pyogenes. I-Retapamulin isebenza ngokuthintela ukwenziwa kweeproteni zebhaktiriya, nto leyo ekhokelela ekuphelisweni kweentsholongwane ezisulelayo kunye nokupheliswa kosulelo lwesikhumba.
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I-Staurosporine, i-streptomyces staurosporeus CAS:62996-74-1
I-Staurosporine yimveliso yendalo ehlukanisiweyo nebhaktheriya iStreptomyces staurosporeus. Ihlelwe njenge-alkaloid enamandla enomsebenzi obalulekileyo webhayoloji, ingakumbi ekuthinteleni ii-protein kinases kunye nokukhuthaza i-apoptosis yeeseli. I-Staurosporine ifundwe ngokubanzi ngenxa yeempawu zayo ze-pharmacological, kubandakanya amandla ayo okulwa nomhlaza kunye nendima yayo njengesixhobo sophando kwizifundo zokubonisa iiseli.
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Ityuwa ye-Phosphomycin disodium CAS:26016-99-9
Ityuwa yePhosphomycin disodium yi-antibiotic ebanzi esetyenziswa kunyango lwezifo ezahlukeneyo zebhaktiriya. Ikwiklasi ye-phosphonic acids kwaye isebenza ngokuthintela ukwenziwa kweeseli zebhaktiriya. Le powder emhlophe ekristale iyanyibilika kakhulu emanzini kwaye idla ngokufakwa ngemithambo okanye ngomlomo. Ityuwa yePhosphomycin disodium yaziwa ngokusebenza kwayo ngokuchasene neebhaktiriya ezahlukeneyo zegram-positive kunye negram-negative, nto leyo eyenza ukuba ibe lukhetho olusebenzisekayo lokunyanga izifo.
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I-Phleomycin CAS:11006-33-0
I-Phleomycin sisibulali-ntsholongwane esinamandla esisetyenziswa kuphando lwebhayoloji yeemolekyuli ekukhetheni iiseli eziqulethe ijini enomdla. Ngomsebenzi obandakanya ukuqhekeka kwe-DNA, i-Phleomycin iyasebenza ngokuchasene neebhaktheriya ezininzi kwaye isetyenzisiwe kakhulu kwizicelo ezahlukeneyo zophando. Le antibiotic isetyenziswa rhoqo kunye nezinye iimpawu zokukhetha ukwenza imigca yeseli ezinzileyo kunye notshintsho olufunekayo lwemfuza. I-Phleomycin ifumaneka kwiifom zolwelo kunye nomgubo, okwenza ukuba ibe lula kwaye ilungele ukuseta okuhlukeneyo kovavanyo. Abaphandi bayayixabisa indlela esebenza ngayo kunye nokuthembeka kwayo ekukhetheni iiseli eziguquliweyo, nto leyo eyenza ukuba ibe sisixhobo esibalulekileyo kwizifundo zobunjineli bemfuza.
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Ityuwa ye-potassium yePenicillin V CAS:132-98-9
Ityuwa ye-potassium ye-Penicillin V yi-antibiotic esetyenziswa ngomlomo ekunyangeni izifo ezibangelwa ziintsholongwane. Iqulethe i-penicillin V, uhlobo lwetyuwa ye-potassium ye-phenoxymethylpenicillin. I-Penicillin V isebenza ngokuphazamisa ukwenziwa kwe-peptidoglycan eludongeni lweseli yebhaktiriya. Oku kwenza buthathaka udonga lweseli kwaye kubulale okanye kuthintele ukukhula kweentsholongwane ezisengozini. Ifumaneka njengeepilisi okanye ii-suspensions ezithathwa ngomlomo ukuze kunyangwe izifo ezibuthathaka ukuya kweziphakathi ngaphandle kwesibhedlele.
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Ityuwa yesodiyam yePenicillin G (ityuwa yesodiyam yeBenzylpenicillin) I-CAS:69-57-8
Ityuwa yesodiyam yePenicillin G yi-antibiotic eyenziwe yi-penicillin G kwimo yayo yetyuwa yesodiyam. Isebenza ngokuthintela ukwenziwa kweengqimba ze-peptidoglycan kwiindonga zeeseli zebhaktiriya, ibulala iibhaktiriya ezisengozini. Ityuwa yesodiyam yePenicillin G ifumaneka njengeekristale ezimhlophe okanye eziphantse zibe mhlophe okanye umgubo ekufuneka uhlanganiswe ube sisicombululo ngaphambi kokuba ufakwe inaliti. Ibonelela ngokuhanjiswa kwe-penicillin G ngendlela ecwangcisiweyo ukunyanga usulelo lweebhaktiriya.
