I-N-(4-Aminobenzoyl)-beta-alanine CAS:7377-8-4
I-N-(4-Aminobenzoyl)-beta-alanine, okanye iProcaine, isetyenziswa kakhulu njengeyeza lokuthomalalisa iintlungu kwiindawo zonyango nezamazinyo. Amandla ayo okuthintela okwethutyana ukuhanjiswa kwemithambo-luvo avumela ukukhululeka kwentlungu ngexesha lotyando oluncinci, unyango lwamazinyo, kunye nokungenelela kolusu. Ngenxa yoko, inceda ekunciphiseni ukungonwabi kunye nokuphucula intuthuzelo yesigulana ngexesha lezi nkqubo. Ukongeza kwiimpawu zayo zokuthomalalisa iintlungu, i-N-(4-Aminobenzoyl)-beta-alanine ifundwe ngemiphumo yayo yonyango ekulawuleni iimeko ezithile zempilo. Uphando lubonisa ukusetyenziswa kwayo kunye namanye amayeza okujongana nentlungu ethile ye-neuropathic, ukubonelela ngokukhululeka kubantu abanesifo seentlungu ezingapheliyo. Ngaphezu koko, le khompawundi ifumene usetyenziso kuphando lovavanyo njengesixhobo sokufunda umsebenzi we-neuronal kunye neempendulo ze-pharmacological. Ukusetyenziswa kwayo kwiindawo zelebhu kwenza izazinzulu ziqonde iinkqubo zokubonisa imiqondiso yemithambo-luvo kwaye ziphande ukusebenzisana kwamayeza kunye neendlela zokusebenza. Ngaphezu koko, i-N-(4-Aminobenzoyl)-beta-alanine ihlolwe ngendima yayo kwiifomyula ezenzelwe iimveliso zokuphelisa iintlungu ezisematheni. Ukufakwa kwayo kwiindlela ezinjalo kujoliswe ekuboneleleni nge-analgesia yendawo kwiintlungu zemisipha, iintlungu zamalungu, kunye nokwenzakala okuncinci, okufaka isandla kwizisombululo ezithengiswa ngaphandle kwemvume kagqirha zokulawula iintlungu ngaphandle kwemiphumo yenkqubo yomzimba. Ngokubanzi, i-N-(4-Aminobenzoyl)-beta-alanine, okanye iProcaine, idlala indima ebalulekileyo kwicandelo lezonyango kunye neyeza njengeyeza lokuthomalalisa iintlungu lasekuhlaleni, inika isiqabu kwiintlungu ngexesha leenkqubo ezahlukeneyo zonyango kunye nonyango lwamazinyo. Ukusetyenziswa kwayo okunokwenzeka konyango ekulawuleni iintlobo ezithile zeentlungu kunye nokusetyenziswa kwayo kuphando kugxininisa ngakumbi ukuguquguquka kwayo kunye nokubaluleka kwayo kuluntu lwezempilo kunye nolwesayensi.
| Ukwakhiwa | N / A |
| Uvavanyo | 99% |
| Inkangeleko | umgubo omhlophe |
| Inombolo ye-CAS | 7377-8-4 |
| Ukupakisha | Encinci kwaye ininzi |
| Beka ubomi kwishelufa | iminyaka eyi-2 |
| Indawo yokugcina izinto | Gcina kwindawo epholileyo neyomileyo |
| Isiqinisekiso | I-ISO. |








