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iimveliso

Iimveliso

I-Pitavastatin CAS:147511-69-1 Umthengisi woMvelisi

I-Pitavastatin sisithinteli se-HMG-CoA reductase esikhuthaza inyathelo lokuqala lokwenziwa kwe-cholesterol. Ibonakala ingenavumba kwaye imhlophe ukuya kumgubo otyheli okhanyayo. Isebenza ngokunciphisa amanqanaba ezinto ezithile ezinamafutha ezifana ne-cholesterol emzimbeni. Ke ngoko, iboniswa ikakhulu kunyango lwe-hypercholesterolaemia kunye nokuthintela izifo zentliziyo. Ayinakunciphisa kuphela i-cholesterol ephezulu kunye ne-triglyceride kwizigulana ezithile, kodwa inokunyusa umxholo we-high density lipoprotein (HDL), amanqanaba e-cholesterol "alungileyo". Kufuneka isetyenziswe ngokubanzi kunye nokutya okufanelekileyo.


Iinkcukacha zeMveliso

Iithegi zeMveliso

Ukusetyenziswa kunye nesiphumo

I-Pivastatin liyeza elilwa ne-hyperlipidemic. Ayisiyo nje kuphela iyeza elitsha, elisebenzayo, elikhuselekileyo, neliyilwe ngamakhemikhali elisekwe kwi-statin elinokusebenza okuphezulu kakhulu, kodwa likwangumthinteli onamandla we-3-hydroxy-3-methylglutaryl CoA (HMG-CoA reductase) reductase. Ayinampembelelo inamandla kuphela ekunciphiseni i-LDL-C kunye ne-TC, kodwa ikwanayo ne-polymorphism ebalulekileyo ye-genetic, i-bioavailability ephezulu, kunye ne-half-life ende. Kwaye bambalwa kuphela abadlula kwi-metabolism ye-CYP2C9. Isetyenziselwa ukunyanga i-primary hyperlipidemia, i-familial hypercholesterolemia, kunye neengxaki ze-lipid ezixutyiweyo.

Isampuli yeMveliso

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图片337(1)

Ukupakisha imveliso:

图片338(1)

Iinkcukacha ezongezelelweyo:

Ukwakhiwa C25H24FNO4
Uvavanyo 99%
Inkangeleko Umgubo omhlophe ukuya kongamhlophe
Inombolo ye-CAS 147511-69-1
Ukupakisha 25KG
Beka ubomi kwishelufa iminyaka eyi-2
Indawo yokugcina izinto Gcina kwindawo epholileyo neyomileyo
Isiqinisekiso I-ISO.

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