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iimveliso

Iimveliso

I-Doxazosin Mesylate CAS: 77883-43-3 Umthengisi woMvelisi

I-Doxazosin mesylate yi-quinazoline compound engumthinteli okhethiweyo we-alpha1 subtype ye-alpha adrenergic receptors. I-Doxazosin mesylate sisizukulwana esitsha se-quinazolone α1 receptor blocker eyenziwe yinkampani yePfizer (e-United States). Inobomi obude obuyihafu, ivelisa iziphumo zayo zokwandisa imithambo yegazi, ukunciphisa ukumelana kwemithambo yegazi kunye nokunciphisa uxinzelelo lwegazi ngokuvala i-a1 receptor. Icetyiswe kwamanye amazwe njengamayeza okuqala eklinikhi okulwa noxinzelelo lwegazi kunye nonyango lwesifo se-prostate.


Iinkcukacha zeMveliso

Iithegi zeMveliso

Ukusetyenziswa kunye nesiphumo

I-Doxazosin mesylate yi-α1 receptor blockers entsha ekhetha kakhulu, enefuthe elikhulu lokubangela ukwehla koxinzelelo lwegazi ngelixa inefuthe elihle lokunciphisa imetabolism ye-lipid. Inganciphisa kakhulu i-serum triglycerides kunye ne-cholesterol iyonke; ikwathintela ngokukhetha i-a1 adrenergic receptor ye-prostate smooth muscle matrix, i-capsule kunye ne-bladder neck, inciphisa iimpawu zezigulane ezine-benign prostatic hyperplasia, inciphise kakhulu ifuthe le-benign prostatic hyperplasia, ngakumbi inefuthe elihle kunyango lwe-dysuria ebangelwa yi-simple prostatic hyperplasia. Inobomi obude obufutshane. Kunokubakho isiyezi, umlomo owomileyo, intloko ebuhlungu, ukubetheka, ukudinwa, iimpawu zincinci, ziyanyamezeleka, ziyanyamalala kwiveki e-1, ngaphandle konyango olukhethekileyo. Akukho hypotension yesimo se-postural eyenzekileyo.

Isampuli yeMveliso

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Ukupakisha imveliso:

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Iinkcukacha ezongezelelweyo:

Ukwakhiwa C24H29N5O8S
Uvavanyo 99%
Inkangeleko Umgubo omhlophe
Inombolo ye-CAS 77883-43-3
Ukupakisha 25KG
Beka ubomi kwishelufa iminyaka eyi-2
Indawo yokugcina izinto Gcina kwindawo epholileyo neyomileyo
Isiqinisekiso I-ISO.

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