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I-2,6-Dichloro-3-nitropyridine CAS:16013-85-7
I-2,6-Dichloro-3-nitropyridine yikhemikhali equlathe ifomula yemolekyuli i-C5H2Cl2N2O2. Yikristale etyheli esetyenziswa kakhulu kwi-organic synthesis kunye nophando lwezamayeza ngenxa yeempawu zayo ezikhethekileyo zekhemikhali. Le khemikhali yaziwa nge-nitro kunye ne-chloro substituents zayo kwiringi ye-pyridine, nto leyo eyenza ukuba ibe luncedo ekuphuhlisweni kweekhompawundi ezahlukeneyo ze-organic.
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I-2,5-Dibromopyrazine CAS:23229-26-7
I-2,5-Dibromopyrazine yikhemikhali ebonakala ngeeathom ezimbini zebromine ezinamathele kwindawo yesibini neyesihlanu yeringi yepyrazine. Olu phawu lolwakhiwo lunika iipropati ezikhethekileyo kwimolekyuli, nto leyo eyenza ukuba ibe luncedo kwiintlobo ngeentlobo zezicelo kuphando nakumashishini.
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I-2-Cyano-3-Chloropyridine CAS:38180-46-0
2-I-Cyano-3-Chloropyridine yikhemikhali enefomula yemolekyuli i-C6H3ClN2. Yinto eqinileyo emthubi okhanyayo esetyenziswa kakhulu kwi-organic synthesis kunye nophando lwezamayeza. Le khemikhali iqulethe iqela le-cyano kunye ne-athomu ye-chlorine eqhotyoshelwe kwiringi ye-pyridine, nto leyo eyenza ukuba ibe luncedo ekuphuhlisweni kweekhompawundi ezahlukeneyo ze-organic ezineempawu ezahlukeneyo.
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I-2-Amino-5-chloropyrazine CAS:33332-29-5
2-I-Amino-5-chloropyrazine yikhemikhali ehlulwe njenge-pyrazine derivative. Iqulethe iqela le-amino kwindawo yesibini kunye ne-athomu ye-chlorine kwindawo yesihlanu yeringi ye-pyrazine. Ulwakhiwo olukhethekileyo lwale khemikhali kunye neempawu zayo zenza ukuba ibe sisakhiwo esibalulekileyo kwi-organic synthesis kunye nophando lweyeza.
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I-2-AMINO-5-BROMO-46-DIMETHYLPYRIDINE CAS:89856-44-0
2-I-Amino-5-Bromo-4,6-Dimethylpyridine yikhemikhali enefomula yemolekyuli i-C8H10BrN2. Yinto eqinileyo emhlophe ukuya kwephuzi esetyenziswa kakhulu kwi-organic synthesis kunye nophando lwezamayeza. Le khompawundi iqulethe iqela le-amino, i-atom ye-bromine, kunye namaqela amabini e-methyl aqhotyoshelwe kwiringi ye-pyridine, nto leyo eyenza ukuba ibe luncedo ekuveliseni iikhompawundi ezahlukeneyo ze-organic ezineempawu ezahlukeneyo.
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I-2-Amino-5-bromopyrazine CAS:59489-71-3
2-I-Amino-5-bromopyrazine yikhemikhali eyinxalenye yosapho lwe-pyrazine, eneqela le-amino kwindawo yesibini kunye ne-athomu ye-bromine kwindawo yesihlanu yeringi ye-pyrazine. Ulwakhiwo olucacileyo lwale khemikhali kunye nokusebenza kwayo kuyenza ibe luncedo kwiindlela ezahlukeneyo zophando kunye noshishino.
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I-3-Methylquinoline CAS: 612-58-8
3-I-Methylquinoline yikhompawundi enuka kamnandi enefomula yemolekyuli i-C10H9N. Lulwelo olungenambala ukuya kolutyheli oluyimbala oluvela kusapho lwe-quinoline lweekhompawundi ze-organic.
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I-2,2,2-Trifluoroethyltrifluoromethanesulfonate CAS:6226-25-1
I-2,2,2-Trifluoroethyltrifluoromethanesulfonate yikhemikhali enefomula yemolekyuli i-C4F9O3S. Isetyenziswa kakhulu njenge-reagent kwi-organic synthesis ngenxa yeempawu zayo ezikhethekileyo zeekhemikhali.
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I-Leupeptin CAS:24125-16-4
ILeupeptin sisithinteli esibuyiselwayo seeproteases esikudidi lweekhompawundi ezaziwa ngokuba zii-protease inhibitors. Isetyenziswa kakhulu kuphando lwebhayoloji kunye nebhayoloji yeeseli ngenxa yokukwazi kwayo ukuthintela uluhlu olubanzi lwee-enzymes zeproteolytic, kubandakanya i-serine, i-cysteine, kunye ne-thiol proteases. ILeupeptin yipowder emhlophe yekristale enyibilikayo emanzini nakwi-organic solvents, nto leyo eyenza ukuba isetyenziswe kwiindawo ezahlukeneyo zovavanyo. Izinzile phantsi kweemeko eziqhelekileyo zokugcina kwaye yaziwa ngokubanzi ngokusebenza kwayo ekukhuseleni iiproteni ekuwohlokeni.
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I-Lomefloxacin hydrochloride CAS:98079-51-7
I-Lomefloxacin hydrochloride luhlobo lwetyuwa ye-lomefloxacin, i-antibiotic ye-fluoroquinolone eyaziwayo ngomsebenzi wayo ngokuchasene neentlobo ezahlukeneyo zeebhaktheriya ezine-Gram-negative kunye nezinye iibhaktheriya ezine-Gram-positive. Le ndlela yongeza ukunyibilika kunye nokuzinza kwe-lomefloxacin, okwenza ifaneleke ukusetyenziswa ngomlomo kunyango lwezifo zebhaktheriya. I-Lomefloxacin hydrochloride isebenza ngokuthintela i-DNA gyrase yebhaktheriya, ngaloo ndlela iphazamisa iinkqubo zokuphindaphinda kwe-DNA kunye nokubhalwa kwe-transcription ezibalulekileyo ekukhuleni kwebhaktheriya. Idla ngokumiselwa kwiintsholongwane zendlela yomchamo, izifo zendlela yokuphefumla, kunye nosulelo lwesikhumba ngenxa yokusebenza kwayo kunye neempawu ezifanelekileyo ze-pharmacokinetic.
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I-Linezolid CAS:165800-03-3
I-Linezolid yi-oxazolidinone antibiotic eyaziwa ngomsebenzi wayo wokulwa neentsholongwane zeGram-positive, kuquka i-methicillin-resistant Staphylococcus aureus (MRSA) kunye ne-vancomycin-resistant enterococci (VRE). Ithintela ukwenziwa kweeproteni zebhaktheriya ngokuzibophelela kwi-23S ribosomal RNA ye-50S subunit, nto leyo ekhokelela kwimiphumo yebhaktheriya okanye yebhaktheriya. I-Linezolid iyafumaneka kwiifomyula zomlomo nezemithambo, nto leyo eyenza ukuba ibe lukhetho oluxabisekileyo lonyango lwezifo zolusu nezezicubu ezithambileyo, i-pneumonia, kunye nezinye izifo ezinzulu zebhaktheriya apho iintlobo ezichaseneyo zixhalabisa khona.
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I-Leupeptin hemisulfate CAS:103476-89-7
I-Leupeptin hemisulfate luhlobo lwetyuwa lwe-leupeptin, i-protease inhibitor eguqulwayo esetyenziswa kakhulu kuphando lwe-biochemical kunye ne-cell biology. Le khompawundi yenziwe ngokukodwa njenge-hemisulfate ukuphucula uzinzo lwayo kunye nokunyibilika kwayo kwizisombululo zamanzi. I-Leupeptin hemisulfate igcina iipropati ezifanayo zokuthintela njenge-leupeptin, ijolise ngempumelelo kwii-enzymes ezahlukeneyo ze-proteolytic ukukhusela iiproteni ekuwohlokeni. Isetyenziswa rhoqo ekucoceni iiproteni, i-cell lysis, kunye novavanyo lomsebenzi we-protease ngenxa yokuthembeka kwayo kunye nokuhambelana kwayo noluhlu lweeprotokholi zovavanyo.
