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Isiseko seHydrocortisone CAS: 50-23-7 Umthengisi woMvelisi
I-Hydrocortisone, 11β,17,21-trihydroxypregn-4-ene-3,20-dione, yeyona GCin iphambili ebantwini bendalo. Nangona kukho inani elikhulu le-GCs zokwenziwa, i-hydrocortisone, ii-esters zayo, kunye neetyuwa zayo zihlala ziyinxalenye ephambili yonyango lwanamhlanje lwe-adrenocortical steroid kunye nomgangatho wokuthelekisa zonke ezinye ii-GC kunye nee-MC. Isetyenziselwa zonke izalathisi ezikhankanyiweyo ngaphambili.
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I-Orlistat CAS: 96829-58-2 Umthengisi woMvelisi
I-Orlistat sisithinteli se-lipase yokugaya ukutya. I-Orlistat yasungulwa e-UK njenge-Xenical yonyango lokutyeba ixesha elide, kungcono ukuba idityaniswe nokutya okune-calories eziphantsi kancinci. I-Orlistat yi-tetrahydro-derivative ye-hypolipaemic lipstatin yendalo (evela kwi-Streptomyces toxyfncini) kwaye inokufumaneka nge-hydrogenation ye-lipstatin okanye ngeendlela ezahlukeneyo zokwenziwa ezibandakanya amanyathelo amaninzi ukusuka kwi-(S) - i-rnalic acid.
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L-Homoarginine Monohydrochloride CAS:1483-01-8 Umthengisi woMvelisi
I-L-Homoarginine sisithinteli se-alkaline phosphatases esingakhuphisaniyo nesikhethekileyo kwi-organism. Le amino acid engabalulekanga ithintela i-alkaline phosphatases yamathambo nesibindi somntu kodwa ayinampembelelo kwi-placental okanye kwi-intestinal isoenzymes. Unyango lwangaphambi konyango nge-L-homoarginine lulibazisa ukukhula kwethumba emzimbeni kwimodeli ye-murine C3H/He osteosarcoma. Ikwathintela ukukhula kwe-pancreatic okubangelwa kukutya okuphezulu kunye nokukhutshwa kwe-enzyme kwiimpuku ezijikelezileyo ze-bile-pancreatic juice, imodeli yokungeniswa kwe-pancreatic enzyme secretion ene-hypercholecystokininemia..
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I-Escitalopram Oxalate CAS:219861-08-2
I-Escitalopram oxalate yi-S-isomer metabolite ye-citalopram kwaye yeyona nto iphambili kumsebenzi wayo wezonyango. Igama layo lekhemikhali yi-(S) -1- [3- (dimethylamino) propyl] -1- (Chemicalbook4-fluorophenyl) -1,3-dihydroisobenzofuran 5-acetonitrile oxalate, Sisithinteli sokubuyisela i-serotonin esikhethiweyo, Inemiphumo emihle yonyango kokubini ukudakumba kwe-endogenous kunye ne-non-endogenous.
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I-Glutathione Encitshisiweyo CAS: 70-18-8 Umthengisi woMvelisi
I-Glutathione (GSH) yi-tripeptide (γ-glutamylcysteinylglycine) esasazeke kakhulu kwizityalo nakwizilwanyana. I-GSH isebenza njenge-nucleophilic co-substrate kwi-glutathione transferases ekususeni i-xenobiotics kwaye ingumnikeli we-electron obalulekileyo kwi-glutathione peroxidases ekunciphiseni i-hydroperoxides. I-GSH ikwabandakanyeka ekuthuthweni kwe-amino acid kunye nokugcinwa kwesimo sokunciphisa i-protein sulfhydryl. Uxinzelelo lwe-GSH luqala kwi-micromolar ezimbalwa kwi-plasma ukuya kwi-millimolar ezininzi kwizicubu ezifana nesibindi.
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Umthengisi weCysteine CAS: 52-90-4
I-L-Cysteine yenye yee-amino acids ezingama-20 zendalo kwaye, ngaphandle kwe-methionine, yeyona kuphela equlethe i-sulfur. Yi-amino acid engeyomfuneko equlethe i-thiol ekhutshwa i-oxidized ukuze yenze i-Cystine. Yi-amino acid engeyomfuneko equlethe i-sulfur ebantwini, enxulumene ne-cystine, i-Cysteine ibalulekile ekuqulunqweni kweproteni, ukususwa kwetyhefu emzimbeni, kunye nemisebenzi eyahlukeneyo ye-metabolic. Ifumaneka kwi-beta-keratin, iproteni ephambili kwiinzipho, ulusu, kunye neenwele, i-Cysteine ibalulekile ekuvelisweni kwe-collagen, kunye nokuqina kwesikhumba kunye nokuthungwa.
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I-Coenzyme A i-asidi yasimahla i-CAS:85-61-0
I-Coenzyme A i-asidi yasimahlayi-cofactor ebalulekileyo esebenza njengomthwali weqela le-acyl kunye neqela elivuselela i-carbonyl kumjikelo we-citric acid kunye ne-fatty acid metabolism. Malunga ne-4% yee-enzymes zeseli zisebenzisa i-CoA njenge-substrate. Yenziwe kwi-pantothenic acid kwinkqubo enamanyathelo ama-5 efuna i-ATP. Inyathelo le-pantothenate kinase lendlela ye-CoA biosynthetic lichongiwe njengenjongo yophuhliso lwee-antibacterial compounds.
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Umthengisi we-Idebenone CAS: 58186-27-9
I-Idebenone yikhompawundi yendalo ephuma kusapho lwe-quinone, efana ne-coenzyme Q-10. Luhlobo lweyeza elenziwe yiTakeda Pharmaceutical Company lokunyanga isifo se-Alzheimer kunye nezinye iziphene zengqondo. Nangona kunjalo, ezi azizange zibe yinkqubela phambili kangako enxulumene nale mpawu. Ngoku ikwasetyenziselwa unyango lwe-Friedreich's ataxia enefuthe elihle kwi-hypertrophy yentliziyo kunye nomsebenzi we-neurological.
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I-Tetracaine Hydrochloride CAS: 136-47-0 Umthengisi woMvelisi
I-Tetracaine hydrochloride yi-benzoate ester. Yi-anesthetic enamandla yendawo efana ne-ester esetyenziselwa i-anesthesia yomphezulu kunye nomqolo. I-Tetracaine hydrochloride liyeza le-anesthetic yendawo kunye ne-ester derivative ye-p-amino benzoic acid. Isebenza ngokuphazamisa ukungena kwee-ion ze-sodium kwiiseli zemithambo-luvo kwaye yenye yezona zinto zisetyenziswa kakhulu kwi-anesthetics zasekhaya.
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I-Leucine CAS: 61-90-5 Umthengisi woMvelisi
ILeucine yenye yee-amino acids ezisibhozo ezibalulekileyo, kwaye ikwii-amino acids ze-aliphatic ngaphakathi kwee-proteins ezingamashumi amabini. I-L-leucine kunye ne-L-isoleucine kunye ne-L-valine zibizwa ngokuba zii-amino acids ezintathu ezine-branched chain. I-L-leucineI-Leucine kunye ne-D-leucine zii-enantiomers. Yikristale emhlophe ekhazimlayo ye-hexahedral okanye umgubo omhlophe wekristale kubushushu begumbi, Ayinavumba, ikrakra kancinci. Xa kukho ii-hydrocarbons, izinzile kwi-aqueous mineral acid. Ngegram nganye inyibilika emanzini angama-40ml kunye ne-acetic acid emalunga ne-100ml. Inyibilika kancinci kwi-ethanol okanye kwi-ether, inyibilika kwi-formic acid, inyibilika i-hydrochloric acid, isisombululo se-alkali hydroxides kunye nesisombululo se-carbonates.
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I-Guanidinopropionic Acid CAS: 353-09-3 Umthengisi woMvelisi
I-Guanidinopropionic acid yikristale emhlophe enyibilika emanzini kwaye iyi-creatine analog. I-Guanidinopropionic acid luhlobo lwee-amino acid derivatives. Yinto ebalulekileyo yekhemikhali eluhlaza kunye nephakathi. Ifumaneka kwi-serum, ebuchosheni, esibindini, kwizintso nakumchamo wezilwanyana ezanyisayo.
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Umthengisi we-Olmesartan CAS:144689-24-7
I-Olmesartan medoxomil,phenyl]phenyl]methyl]imidazole-4-carboxylate (iBenicar, i-Olmetec) isebenzisa inkqubo ye-tetrazolering njengenkqubo yayo ye-asidi, ethatha inxaxheba ekubopheni ii-receptor. Xa inikwa isigulane, iyeza lisebenza ngokukhawuleza nangokupheleleyo yi-ester hydrolysis ye-medoxomil ngexesha lokufunxwa kwindlela yesisu. I-Olmesartan yi-biphenylyltetrazole. Inendima njenge-arhente yokulwa noxinzelelo lwegazi kunye ne-angiotensin receptor antagonist.
