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Umthengisi weTert-Butylamine CAS: 75-64-9
I-Tert-butylamine yi-amine ephambili ye-aliphatic eyi-ethylamine ethathelwe indawo ngamaqela amabini e-methyl kwindawo yoku-1. Yisiseko esidibeneyo se-tert-butylammonium. I-Tert-Butylamine ikwasetyenziselwa ukuvelisa amayeza okubulala ukhula, oko kukuthi, i-terbacil kunye ne-triazines terbutylazine, i-terbumeton, kunye ne-terbutryn kunye ne-insecticides (umz., i-diafenthiuron). I-derivative ikwacetywayo njengesiqinisi sezinto zokuthambisa.
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Umthengisi weLysine HCL CAS: 657-27-2
I-Lysine HCLyi-amino acid ebalulekileyo kwizilwanyana nakubantu. I-L-Lysine iyimfuneko ekuvelisweni kweproteni emzimbeni nasekukhuleni kakuhle. I-L-lysine yehlisa amanqanaba e-cholesterol ngokuvelisa i-carnitine. I-L-lysine inceda ekufunxweni kwe-calcium, i-zinc kunye ne-iron. Abadlali basebenzisa i-L-lysine njengesongezelelo sokwakha ubunzima obuncinci kunye nempilo efanelekileyo yemisipha namathambo. I-L-lysine ikhuphisana ne-arginine ngexesha lokuzala kwentsholongwane kwaye inciphisa usulelo lwe-herpes simplex virus. Ukongezwa kwe-L-lysine kunciphisa ixhala elingapheliyo ebantwini. I-Lysine inciphisa i-viscosity yesisombululo se-serum albumin xa kujovwa.
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I-Griseofulvin CAS:126-07-8 Umthengisi woMvelisi
I-Griseofulvin yi-antibacterial elwa ne-antifungal engeyiyo i-polyene class; inokuthintela kakhulu i-mitosis yeseli yefungus kwaye iphazamise ukwenziwa kwe-DNA yefungus; ingakwazi nokubophelela kwi-tubulin ukuthintela ukwahlukana kweeseli zefungus. Isetyenziswe kumayeza eklinikhi ukususela ngo-1958 kwaye okwangoku isetyenziswa kakhulu ekunyangeni usulelo lwefungus lwesikhumba kunye ne-stratum corneum enefuthe elinamandla lokuthintela kwi-Trichophyton rubrum kunye ne-Trichophyton tonsorans, njl. I-Griseofulvin ayisiyo-antibiotic esetyenziswa kakhulu kuphela kunyango lwezonyango lwesulelo lwefungus lwesikhumba kunye ne-cuticle, kodwa ikwasetyenziswa kwezolimo ukuthintela nokunyanga izifo zefungus; umzekelo, inamandla akhethekileyo ekunyangeni uhlobo lwe-candidiasis kwi-apile enokubangela usulelo ngexesha lokuvuna.
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Umthengisi we-Olmesartan Medoxomil CAS:144689-63-4
I-Olmesartan Medoxomil, sisixhobo esitsha esikhethiweyo nesikhuphisanayo se-angiotensin II type 1 receptor antagonist kwaye sithintela ngamandla iimpendulo ze-Ang.ll-induced pressor. Esi sidakamizwa sithintele ngokukhuphisana ukubopha [125I1]-All kwi-AT1 receptors kwi-bovine adrenal cortical membranes, kodwa asizange sibe nefuthe ekubopheni kwi-AT2 receptors kwi-bovine cerebellar membranes. I-Olmesartan medoxomil ikwabonakalisiwe ukuba inciphisa uxinzelelo lwegazi ngokufanelekileyo kakhulu kune-losartan kunye ne-ACE inhibitor captopril kwaye ngokufanelekileyo njenge-pbloker atenolol.
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Umthengisi we-L-Citrulline Malate (2:1) CAS: 70796-17-7
I-L-Citrulline Malate (2:1)yi-compound equlathe iCitrulline, i-amino acid engabalulekanga efumaneka kakhulu kwiimelon, kunye ne-malate, into ephuma kwi-apile. Kakade ke, ukuze ufumane iCitrulline neMalate eyaneleyo ukuze ufumane iingenelo zayo zokuphucula ukusebenza kuya kufuneka utye ii-watermelon ezininzi kunye nama-apile mhlawumbi ungagula, kodwa uyayibona ingongoma yam. I-Citrulline Malate isetyenziswe ngempumelelo enkulu ngoogqirha baseYurophu abaye baxela iziphumo zamandla anyukileyo kunye neemvakalelo zempilo iyonke.
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Umthengisi woMvelisi weDuloxetine HCL CAS:136434-34-9
I-Duloxetine HCLyi-serotonin ekhethiweyo (5-HT) kunye ne-norepinephrine reuptake inhibitor (SSNRI) yokusetyenziswa ngomlomo, kwaye okwangoku ivunyiwe e-US naseYurophu kunyango lwe-major depression disorder (MDD) kunye ne-diabetes peripheral neuropathic pain (DPN).
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Umthengisi weMinoxidil Sulfate CAS: 83701-22-8
I-Minoxidil sulfate (MXS) sisithako esiphuma kwi-minoxidil. Inokunyibilika kakhulu emanzini kwaye ingumdibanisi onamandla. I-MXS inamandla okunyanga i-androgenic alopecia okanye i-paldness yamadoda. I-ATP-sensitive potassium channel opener ekhethiweyo. Yi-metabolite esebenzayo ye-minoxidil kwaye inamandla (IC50 = 0.14) vascular smooth muscle relaxant.
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I-R(+)-Alpha Lipoic Acid Sodium Salt CAS:176110-81-9
Ityuwa yeSodium ye-R(+)-Alpha Lipoic Acidyi-enzyme eveliswa ngumzimba womntu ngokwendalo. Ithatha inxaxheba kwi-aerobic metabolism ukuvelisa amandla. Ikwayi-antioxidant enamandla enokususa ii-free radicals ezibangela ukwaluphala okukhawulezileyo kunye nezifo. I-lipoic acid yahlulwe yaba yi-L-lipoic acid, i-dextro-lipoic acid kunye ne-mixed lipoic acid. Phakathi kwazo, i-dexlipoic acid ibonakalisiwe ukuba inokufumaneka kakuhle kwezinto eziphilayo, uzinzo, kwaye ibonelela ngeenzuzo ezahlukeneyo zempilo.
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I-Cysteine HCL Anhydrous CAS: 52-89-1 Umthengisi woMvelisi
I-Cysteine HCL Engenamanziyi-hydrochloride efunyenwe ngokudibanisa i-L-cysteine kunye ne-molar equivalent enye ye-hydrogen chloride. Inendima njenge-EC 4.3. 1.3 (histidine ammonia-lyase) inhibitor, iarhente yonyango lomgubo kunye ne-metabolite yomntu. Iqulethe i-L-cysteinium.
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I-L-Arginine Alpha-Ketoglutarate(1:1) I-CAS:16856-18-1
I-L-Arginine Alpha-Ketoglutarate,okanye i-AAKG. Iqulethe i-L-arginine, i-amino acid ebalulekileyo eveliswa yimizimba yethu ngokwendalo. Ikwanayo ne-A-ketoglutarate, imolekyuli esebenza ngeendlela ezininzi ekwaveliswa emzimbeni. I-Arginine alpha-ketoglutarate sisongezelelo sokutya esiqulathe i-amino acid arginine isakhiwo seprotheyini kunye ne-alpha-ketoglurate, ikhompawundi eqhekeza iiswekile kunye nee-amino acids. Zombini izinto ze-AAKG zinemisebenzi eyahlukeneyo kwaye zinokubonelela ngeenzuzo.
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I-Clascoterone CAS:19608-29-8 Umthengisi woMvelisi
I-Clascoterone sisithinteli se-androgen receptor esiphuhliswa njengekhrimu kunye nesisombululo se-topical yiCassiopea (inkampani yeCosmo Pharmaceuticals) yokunyanga iingxaki zesikhumba ezixhomekeke kwi-androgen, kubandakanya i-androgenetic alopecia kunye ne-acne vulgaris. Nangona indlela echanekileyo yokusebenza kwe-clascoterone kunyango lwe-acne vulgaris ingaziwayo, eli yeza kukholelwa ukuba likhuphisana ne-androgen dihydrotestosterone yokubopha kwi-androgen receptors kwi-sebaceous gland kunye ne-hair follicles ukunciphisa imiqondiso efunekayo kwi-acne pathogenesis.
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I-Pitavastatin CAS:147511-69-1 Umthengisi woMvelisi
I-Pitavastatin sisithinteli se-HMG-CoA reductase esikhuthaza inyathelo lokuqala lokwenziwa kwe-cholesterol. Ibonakala ingenavumba kwaye imhlophe ukuya kumgubo otyheli okhanyayo. Isebenza ngokunciphisa amanqanaba ezinto ezithile ezinamafutha ezifana ne-cholesterol emzimbeni. Ke ngoko, iboniswa ikakhulu kunyango lwe-hypercholesterolaemia kunye nokuthintela izifo zentliziyo. Ayinakunciphisa kuphela i-cholesterol ephezulu kunye ne-triglyceride kwizigulana ezithile, kodwa inokunyusa umxholo we-high density lipoprotein (HDL), amanqanaba e-cholesterol "alungileyo". Kufuneka isetyenziswe ngokubanzi kunye nokutya okufanelekileyo.
