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I-β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Salt CAS:24292-60-2
β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Saltyi-coenzyme esasazeke kakhulu kwizinto eziphilayo, Ithatha inxaxheba kwiimpendulo zokunciphisa i-oxidation. Isebenza njengomthwali we-electron kwiimpendulo ezininzi, i-oxidized alternately (NADP+) kwaye incitshiswe (NADPH).β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Saltsisithako apho i-nicotinic acid amide adenine dinucleotide kunye nemolekyuli ye-phosphate zibotshelelwe yi-ester bond. Yi-hydrogen receptor kwaye ingasetyenziselwa uphuhliso kunye nophuhliso lwee-reagents ezahlukeneyo zokuxilonga kwi-in vitro.
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I-β-Nicotinamide Adenine Dinucleotide Ityuwa yeLithium (ityuwa ye-NAD Lithium) CAS:64417-72-7
β-Nicotinamide Adenine Dinucleotide Ityuwa yeLithiumyi-coenzyme ephambili kwimetabolism. Ifumaneka kuzo zonke iiseli eziphilayo, i-NAD ibizwa ngokuba yi-dinucleotide kuba inee-nucleotides ezimbini ezidityaniswe ngamaqela azo e-phosphate. I-nucleotide enye iqulethe i-adenine nucleobase kwaye enye i-nicotinamide. I-NAD ikhona ngeendlela ezimbini: ifom e-oxidized kunye ne-reduced, efinyeziweyo njenge-NAD+ kunye ne-NADH (H ye-hydrogen), ngokulandelanayo.
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I-Venlafaxine CAS:93413-69-5
IVenlafaxine sisithomalalisi sokudakumba seklasi ye-serotonin kunye ne-norepinephrine reuptake inhibitor (SNRI). Eli yeza laqalwa ukuphuhliswa nguWyeth kwi-19Chemicalbook93 kwaye ngoku lithengiswa yiPfizer. Eli yeza livunyiwe ukunyanga isifo sokudakumba esikhulu (MDD), isifo sokudakumba esiqhelekileyo (GAD), kunye nokudakumba okunxulunyaniswa nexhala.
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Umthengisi weCiclopirox Ethanolamine CAS:41621-49-2
I-Ciclopirox ethanolamine sisithako esibanzi sokulwa ne-gfungal, ikwabonisa umsebenzi wokulwa neentsholongwane kwiintsholongwane ezininzi ze-Gram-positive kunye ne-Gram-negative, kwaye ineempawu zokulwa nokuvuvukala. Isetyenziswa njengonyango lwesikhumba kunye nosulelo lwezipikili.
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Desvenlafaxine Succinate CAS:386750-22-7
I-Desvenlafaxine Succinate yi-dual serotonin kunye ne-norepinephrine reuptake inhibitor (SNRI) eyavunywayo kunyango lwe-major depression disorder (MDD) e-United States ngo-2008. Ukuze kuphuculwe ukusebenza kakuhle kunye neprofayili yokhuseleko lwe-venlafaxine, uWyeth wafumanisa waza waphuhlisa enye yee-metabolites eziphambili ze-venlafaxine, oko kukuthi i-O-desmethyl metabolite (desvenlafaxine).
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I-Doxazosin Mesylate CAS: 77883-43-3 Umthengisi woMvelisi
I-Doxazosin mesylate yi-quinazoline compound engumthinteli okhethiweyo we-alpha1 subtype ye-alpha adrenergic receptors. I-Doxazosin mesylate sisizukulwana esitsha se-quinazolone α1 receptor blocker eyenziwe yinkampani yePfizer (e-United States). Inobomi obude obuyihafu, ivelisa iziphumo zayo zokwandisa imithambo yegazi, ukunciphisa ukumelana kwemithambo yegazi kunye nokunciphisa uxinzelelo lwegazi ngokuvala i-a1 receptor. Icetyiswe kwamanye amazwe njengamayeza okuqala eklinikhi okulwa noxinzelelo lwegazi kunye nonyango lwesifo se-prostate.
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Umthengisi we-L-Isoleucine CAS: 73-32-5
I-L-Isoleucine, eyaziwa ngokuba yi-Isoleucine, yi-amino acid eyi-isomer ye-leucine. Ibalulekile ekuqulunqweni kwe-hemoglobin kunye nokulawula amanqanaba eswekile yegazi kunye namandla. I-L-Isoleucine yi-isomer ye-L-leucine kwaye yi-amino acid ebalulekileyo. Yenziwe kwi-threonine kwaye yi-amino acid ye-hydrophobic.
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Umthengisi weCaptopril CAS: 62571-86-2
I-Captopril yeyona ifundwa kakhulu kwii-angiotensin-converting enzyme inhibitors ezicetywayo njengeyeza lokulwa noxinzelelo lwegazi. Ithintela i-angiotensin-converting enzyme, ethintela ukwakheka kwe-angiotensin II kwaye inciphise impembelelo yayo yokuvaleka kwegazi kwimithambo yegazi kunye nemithambo yegazi. Uxinzelelo olupheleleyo lwemithambo yegazi luyancitshiswa, nto leyo ekhokelela ekunciphiseni uxinzelelo lwemithambo yegazi.
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Umthengisi woMvelisi weCandesartan CAS:139481-59-7
I-Candesartan yi-angiotensin II receptor I (AT1) antagonist, i-IC50s=1.12 kunye ne-2.86 nM ye-bovine adrenal cortex kunye ne-rabbit aorta ngokwahlukeneyo. Ithintela ngokukhetha ukucutheka okubangelwa yi-angiotensin II kwi-rabbit aortic strips ngaphandle kwefuthe ekucuthekeni okubangelwa zezinye izinto ezifana ne-norepinephrine, i-KCl, i-serotonin, i-PGF2α okanye i-endothelin.
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I-Candesartana Cilexetila CAS:145040-37-5
ICendesartan Celexetil yi-ester analog ye-angiotensin II antagonist ICendesartan (sc-217825). Ukuchasana kwale receptor kuthintela ukubopha kwe-angiotensin II, i-vasoconstrictor enamandla. Oku kunefuthe elipheleleyo lokusasazeka kwemithambo yegazi kunye nomthamo wegazi onyukayo. ICendesartan Celexetil Ester sisithinteli se-AT1.
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Umthengisi weBupropion CAS: 34911-55-2
I-Bupropion yi-aromatic ketone eyi-propiophenone ephethe iqela le-tert-butylamino kwindawo yesi-2 kunye ne-chloro substituent kwindawo yesi-3 kwiringi ye-phenyl. Inendima njenge-antidepressant, i-contaminant yokusingqongileyo kunye ne-xenobiotic. Yi-amino compound yesibini, ilungu le-monochlorobenzenes kunye ne-aromatic ketone.
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Umthengisi weBezafibrate CAS:41859-67-0
I-Bezafibrate yi-monocarboxylic acid amide efunyenwe ngokudityaniswa okusemthethweni kweqela le-carboxy le-4-chlorobenzoic acid kunye neqela le-amino le-2-[4-(2-aminoethyl)phenoxy]-2-methylpropanoic acid. I-Benafibrate isetyenziselwa unyango lwe-hyperlipidaemia. Inendima njenge-xenobiotic, isingcolisi sendalo, i-geroprotector kunye neyeza lokulwa ne-lipidemic. Yi-monocarboxylic acid, i-aromatic ether, ilungu le-monochlorobenzenes kunye ne-monocarboxylic acid amide. Inxulumene ngokusebenzayo ne-propionic acid.
